4.10.15

AMOXILLIN

antibacterial (penicillin class)


Brands/Synonyms , Amoxi-Tabs, Amoxident, Amoxil, Amoxycillin,Amoram, Amoxsan

 Amoxi, Amoxi-Drops, Amoxi-Inject DisperMox, Galenamox, Moxatag

Therapeutics

Interactions

Synergistic antibacterial effect with aminoglycosides (but not synergistic for adverse/toxic effects)
Avoid coadministration with doxycycline, because doxycycline reduces cell protein synthesis required for formation of cell walls, the substrate on which penicillins act (i.e., coadministration predisposes to treatment failure)

Soundalike Alert

Ampicillin
Amoxicillin-clavulanic acid

Available Formulations

Tab
50, 100, 200, 250, 400, 500 mg
Cap
250, 500 mg
Oral solution
25, 50 mg/mL

Indications

Dog
Gram-positive aerobic bacterial infections (e.g., pyoderma)
10-20
mg/kg PO q 12h
Dog
Leptospirosis
22
mg/kg PO q 8h
Dog
Helicobacteriosis
50
mg/kg PO q 12h
Cat
Cat bite abscesses
11-22
mg/kg PO q 12h
Cat
Helicobacteriosis
20
mg/kg PO q 12h


Precautions

Contraindications

Hypersensitivity to the drug, both humans handling the drug (penicillin allergy) and animals receiving it
Resistant infections (common: 6% rate of single drug resistance and 28% rate of multidrug resistance including amoxicillin for E. coli infections in dogs)
Ineffective for borreliosis/Lyme disease
Lack of benefit in feline upper respiratory infection

Adverse Side Effects

Occasional anorexia, inappetence, vomiting, which resolve with discontinuation of the drug
Fanconi syndrome associated with amoxicillin treatment in a dog
Among the lowest reported rate of adverse effects (7.5%) for antibacterials according to owner surveys

Teratogenicity/Pregnancy/Lactation

Rodent studies suggest amoxicillin is generally safe in pregnancy and lactation



Pearls

Example of rate of bacterial resistance: 33% (130/396) of E. coli infections in dogs are 
resistant to amoxicillin
Renal excretion means heightened concentration of amoxicillin in urine, disproportionately 
more effective for bacterial cystitis
Endotoxemia reduces elimination by 2- to 3-fold in dogs; consider longer interdose interval 
if sepsis is suspected
Food, water reduce absorption of amoxicillin, but all tablets should be followed by an oral 
dose of water (and/or for practical reasons of compliance for many owners, a small treat) 
to ensure passage to the stomach
Oral amoxillin has far superior absorption compared to oral ampicillin
Anecdotal reports of greater incidence of immune-mediated hemolytic anemia in animals
treated with beta-lactam antibacterials like amoxicillin; judicious use of such 
antibacterials is recommended in general and in these patients in particular


References

PubMed – 20102505
PubMed – 8968890
PubMed – 18539493
PubMed – 7820765


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